ActiTide-AH3(Liquefied 500) / Acetyl hexapeptide-8

Inkcazelo emfutshane:

Imveliso yepeptide inezona zicelo zibanzi zokuchasa imibimbi. Ukunciphisa ubunzulu bemibimbi ebangelwa kukucutheka kwezihlunu zobuso ingakumbi ebunzi nakwikona yamehlo. Enye indlela ekhuselekileyo, engabizi kakhulu, ethambileyo yeBotox, ngakumbi ijolise kwisiphumo sendlela yokwenza imibimbi ngendlela ekhethekileyo.

Umxholo wepeptide we-ActiTide-AH3 (Liquefied 500) yi-500ppm.


Iinkcukacha zeMveliso

Iithegi zeMveliso

Igama lebrand ActiTide-AH3(Liquefied 500)
Inombolo yeCAS. 7732-18-5; 616204-22-9; 1117-86-8
INCI Igama Amanzi; I-Acetyl hexapeptide-8; Caprylyl glycol
Isicelo I-Lotion, iiSerum, iMask, isicoci sobuso
Iphakheji 1kg/ibhotile
Imbonakalo Ulwelo olucacileyo noluselubala
Umxholo wePeptide 0.045 - 0.060%
Ukunyibilika Amanzi anyibilikayo
Umsebenzi Peptide series
Beka ubomi kwishelufa iminyaka eyi-2
Ugcino Gcina kwindawo epholileyo neyomileyo, kude nokukhanya. 2 ~ 8°C yokugcina
Umthamo 3.0-10.0%

Isicelo

Uphando kwiindlela ezisisiseko zokulwa nemibimbi lukhokelele ekufunyanweni kwe-ActiTide-AH3, i-hexapeptide entsha ephuhliswe ngendlela yenzululwazi ukusuka kuyilo oluqiqileyo ukuya kwimveliso ye-GMP, eneziphumo ezilungileyo.

I-ActiTide-AH3 ihambisa ukusebenza kakuhle kokunciphisa imibimbi ngokuthelekiswa ne-Botulinum Toxin Type A, ngelixa ikhusela umngcipheko wokutofa kunye nokubonelela ngeendleko eziphezulu.

Izibonelelo zokuthambisa:
I-ActiTide-AH3 inciphisa ubunzulu bokushwabana okubangelwa kukufinyaniswa kwemisipha yobuso, kunye neziphumo ezivakalayo kwibunzi kunye nemibimbi yeperiocular.

Indlela yokwenza:
Ukucutheka kwezihlunu kwenzeka ekukhutshweni kwe-neurotransmitter kwi-synaptic vesicles. I-SNARE complex - indibano ye-ternary ye-VAMP, i-Syntaxin, kunye ne-SNAP-25 iiprotheni - ibalulekile kwi-vesicle docking kunye ne-neurotransmitter exocytosis (A. Ferrer Montiel et al., JBC 1997, 272: 2634-2638). Olu bunzima lusebenza njenge-hook yeselula, ukubamba i-vesicles kunye nokuqhuba i-membrane fusion.

Njengomfanekiso wesakhiwo se-SNAP-25 N-terminus, i-ActiTide-AH3 ikhuphisana ne-SNAP-25 yokufakwa kwi-SNARE complex, imodareyitha indibano yayo. Ukuchithwa kwe-SNARE eyinkimbinkimbi yonakalisa i-vesicle docking kunye nokukhululwa kwe-neurotransmitter elandelayo, okukhokelela ekunciphiseni ukunyanzeliswa kwemisipha kunye nokuthintela imibimbi kunye nokuqulunqwa komgca ococekileyo.

I-ActiTide-AH3 yindlela ekhuselekileyo, eyongayo, kwaye ethambileyo kune-Botulinum Toxin Type A. Ijolise ngokwesihloko kwindlela yokubumba imibimbi kodwa isebenza ngendlela eyahlukileyo.


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